Expertise Cloud

Agave sisalanaAnticancerBenzylidene acetalbetamethasoneBF3.OEt2Biological activitydehydrogenationD-glucosed-Mannoseepoxidationfive componentFURANONE-COUMARINSGanodermagas chromatography–mass spectroscopy (GC-MS)glucose effectgorgonianGrignardGrignard reactionH1N1H5N1hecogeninhomogeneous catalysisHorner-Wadsworth-Emmons reactionhuman Topoisomerase IIhydrolysisHypoglycemic effectIC50immunityin vitro studyInhibitorINHIBITORSironisagarinisoquinolinesisoquinolinonesIsothermalisozymeKB)Knoevenagel condensationlaccaseLEAVESLeptogorgia sarmentosaLewis acidMannosemarine organismsmenisporopsin AMenisporopsis theobromaeMetabolic syndromemetal-mediated domino reactionminimum inhibitory concentrationsmolecular dockingmolecular dynamicsmolecular modelingMOLECULAR-BASISmulticomponent reactionsNaphthaquinone aliphatic amideNaphthaquinone aliphatic esternaphtholNaphthoquinonenaphthoquinone esterNAPHTHOQUINONE ESTERSNaphthoquinonesNATURAL-PRODUCTSNClN-formylnornuciferinenonhumanoseltamivirOseltamivir phosphatepalladiumPatchoulipatchouli (Pogostemon cablin)patchouli alcohol (patchoulol)pentylidene ketalpentylidine acetalPeptidomimeticpeptidomimetic agentPEXELPinostrobinPlasmepsin VPlasmodium falciparumPLASMODIUM-FALCIPARUMPogostemon cablinpolyketide synthasePolyoxygenated cholestanesPolypropylenereductive ring openingselective ring openingsteroidssynthesisTamifluการเปิดวงคีทัลการสังเคราะห์ไข้หวัด2009ไข้หวัดนกทามิฟลูทามิฟอสเฟอร์น้ำตาลโมเลกุลเดี่ยวบอระเพ็ดแมนโนสโอเซลทามิเวียร์

Interest


Administrative Profile


    Resource


    งานวิจัยในรอบ 5 ปี

    Project

    งานวิจัยที่อยู่ระหว่างการดำเนินการ
    • ทุนใน 6 โครงการ (ที่ปรึกษาโครงการ 4 โครงการ, ผู้ร่วมวิจัย 2 โครงการ)
    • ทุนนอก 0 โครงการ
    งานวิจัยที่เสร็จสิ้นแล้ว
    • ทุนใน 16 โครงการ (หัวหน้าโครงการ 5 โครงการ, ผู้ร่วมวิจัย 11 โครงการ)
    • ทุนนอก 14 โครงการ (หัวหน้าโครงการ 7 โครงการ, ที่ปรึกษาโครงการ 1 โครงการ, ผู้ร่วมวิจัย 6 โครงการ)

    แนวโน้มผลงานทั้งหมดเทียบกับแนวโน้มผลงานในรอบ 5 ปี

    Output

    • บทความ 83 เรื่อง (ตีพิมพ์ในวารสารวิชาการ 49 เรื่อง, นำเสนอในการประชุม/สัมมนา 34 เรื่อง)
    • ทรัพย์สินทางปัญญา 4 เรื่อง (อนุสิทธิบัตร 2 เรื่อง, สิทธิบัตร 2 เรื่อง)

    แนวโน้มการนำผลงานไปใช้ประโยชน์ในด้านต่างๆ

    Outcome

    • การนำผลงานไปใช้ประโยชน์ 16 เรื่อง (เชิงวิชาการ 12 เรื่อง, เชิงนโยบาย/บริหาร 0 เรื่อง, เชิงสาธารณะ 4 เรื่อง, เชิงพาณิชย์ 0 เรื่อง)

    รางวัลที่ได้รับ

    Award

    • รางวัลที่ได้รับ 7 เรื่อง (ประกาศเกียรติคุณ/รางวัลนักวิจัย 1 เรื่อง, รางวัลผลงานวิจัย/สิ่งประดิษฐ์ 5 เรื่อง, รางวัลผลงานนำเสนอในการประชุมวิชาการ 1 เรื่อง)

    นักวิจัยที่มีผลงานงานร่วมกันมากที่สุด 10 คนแรก


    Scopus h-index

    #Document titleAuthorsYearSourceCited by
    1Transforming rhinacanthin analogues from potent anticancer agents into potent antimalarial agentsKongkathip N., Pradidphol N., Hasitapan K., Grigg R., Kao W., Hunte C., Fisher N., Warman A., Biagini G., Kongsaeree P., Chuawong P., Kongkathip B.2010Journal of Medicinal Chemistry
    53(3),pp. 1211-1221
    26
    2Palladium catalysed reaction of allene with phenols. Phenoxymethyl-1,3-dienes and their further reactionsGrigg R., Kongkathip N., Kongkathip B., Luangkamin S., Dondas H.2001Tetrahedron
    57(37),pp. 7965-7978
    26
    3Short step synthesis of 1,3-dimethyl-2,9-dioxabicyclo [3.3.1] nonane: An insect attractant.Kongkathip B., Kongkathip N.1984Tetrahedron Letters
    25(20),pp. 2175-2176
    25
    4Development of patchouli extraction with quality control and isolation of active compounds with antibacterial activityKongkathip N., Pornpat S., Kongkathip B., Pankaew Y., Tanasotnbat M., Udomkusonsri P.2009Kasetsart Journal - Natural Science
    43(3),pp. 519-525
    23
    5Synthesis of novel naphthoquinone aliphatic amides and esters and their anticancer evaluationKongkathip B., Akkarasamiyo S., Hasitapan K., Sittikul P., Boonyalai N., Kongkathip N.2013European Journal of Medicinal Chemistry
    60,pp. 271-284
    20
    6A new and efficient asymmetric synthesis of oseltamivir phosphate (Tamiflu) from D-glucoseKongkathip B., Akkarasamiyo S., Kongkathip N.2015Tetrahedron
    71(16),pp. 2393-2399
    19
    7Novel laccases of Ganoderma sp. KU-Alk4, regulated by different glucose concentration in alkaline mediaTeerapatsakul C., Abe N., Bucke C., Kongkathip N., Jareonkitmongkol S., Chitradon L.2007World Journal of Microbiology and Biotechnology
    23(11),pp. 1559-1567
    19
    8First synthesis of 3,16,20-polyoxygenated cholestanes, new cytotoxic steroids from the gorgonian Leptogorgia sarmentosaBoonananwong S., Kongkathip B., Kongkathip N.2008Steroids
    73(11),pp. 1123-1127
    18
    9Pinostrobin from Boesenbergia pandurata Is an inhibitor of Ca 2+-Signal-Mediated Cell-Cycle regulation in the Yeast Saccharomyces cerevisiaeWangkangwan W., Boonkerd S., Chavasiri W., Sukapirom K., Pattanapanyasat K., Kongkathip N., Miyakawa T., Miyakawa T.2009Bioscience, Biotechnology and Biochemistry
    73(7),pp. 1679-1682
    17
    10Stereospecific total synthesis of amberketal and a homologueKongkathip B., Kongkathip N., Janthorn S., Virarangsiyakorn D.1999Chemistry Letters
    (1),pp. 51-52
    17
    11Synthesis of betamethasone from the waste of Thai Agave sisalanaKongkathip N., Kongkathip B., Noimai N.2006Synthetic Communications
    36(7),pp. 865-874
    16
    12Catalytic processes for the functionalisation and desymmetrisation of malononitrile derivativesGrigg R., Hasakunpaisarn A., Kilner C., Kongkathip B., Kongkathip N., Pettman A., Sridharan V.2005Tetrahedron
    61(39),pp. 9356-9367
    16
    13A facile palladium catalysed 3-component cascade route to functionalised isoquinolinones and isoquinolinesGrigg R., Elboray E.E., Elboray E.E., Akkarasamiyo S., Akkarasamiyo S., Chuanopparat N., Chuanopparat N., Dondas H.A., Abbas-Temirek H.H., Fishwick C.W.G., Aly M.F., Kongkathip B., Kongkathip N.2016Chemical Communications
    52(1),pp. 164-166
    14
    14Stereoselective pd(0) catalysed five component cascade synthesis of complex z, z-bisallylaminesGrigg R., Akkarasamiyo S., Akkarasamiyo S., Chuanopparat N., Chuanopparat N., Elboray E.E., Elboray E.E., Aly M.F., Abbas-Temirek H.H., Kongkathip B., Kongkathip N.2013Chemical Communications
    49(20),pp. 2007-2009
    14
    15A concise and practical synthesis of oseltamivir phosphate(Tamiflu) from d-mannoseChuanopparat N., Kongkathip N., Kongkathip B.2012Tetrahedron
    68(34),pp. 6803-6809
    14
    16Further study on synthesis and evaluation of 3,16,20-polyoxygenated steroids of marine origin and their analogs as potent cytotoxic agentsBunyathaworn P., Boonananwong S., Kongkathip B., Kongkathip N.2010Steroids
    75(6),pp. 432-444
    13
    17A Novel Synthetic Approach from Diosgenin to a 17α-Hydroxy Orthoester via a Regio- and Stereo-Specific Rearrangement of an Epoxy EsterChaosuancharoen N., Kongkathip N., Kongkathip B.2004Synthetic Communications
    34(6),pp. 961-983
    12
    18Inhibitory effects of 2-substituted-1-naphthol derivatives on cyclooxygenase I and IIKongkathip B., Sangma C., Kirtikara K., Luangkamin S., Hasitapan K., Jongkon N., Hannongbua S., Kongkathip N.2005Bioorganic and Medicinal Chemistry
    13(6),pp. 2167-2175
    11
    19Synthesis of cytotoxic novel 9,11-secosterol analogs: Structure/activity studiesKongkathip B., Hasakunpaisarn A., Boonananwong S., Kongkathip N.2010Steroids
    75(12),pp. 834-847
    11
    20A new and efficient asymmetric synthesis of oseltamivir phosphate(Tamiflu) from D-mannoseChuanopparat N., Kongkathip N., Kongkathip B.2012Tetrahedron Letters
    53(46),pp. 6209-6211
    10
    21Immunological and bactericidal effects of turmeric (Curcuma longa Linn.) extract in pacific white shrimps (Litopenaeus vannamei Boone)Vanichkul K., Areechon N., Kongkathip N., Srisapoome P., Chuchird N.2010Kasetsart Journal - Natural Science
    44(5),pp. 850-858
    9
    22Synthesis of isagarin, a tetracyclic naphthoquinone via a palladium-catalyzed cyclizationPloysuk C., Kongkathip B., Kongkathip N.2007Synthetic Communications
    37(9),pp. 1463-1471
    9
    23FeCl3-catalysed cleavage of 1,2-butanediacetal protected diolsTzschucke C., Pradidphol N., Diéguez-Vázquez A., Kongkathip B., Kongkathip N., Ley S.2008Synlett
    (9),pp. 1293-1296
    8
    24Regioselective ring opening of exo- and endo-3,4-benzylidene acetals of arabinopyranoside derivatives with Lewis acids and reducing agentsRujirawanich J., Kongkathip B., Kongkathip N.2011Carbohydrate Research
    346(7),pp. 927-932
    7
    25Determination of a pyranocoumarin and three carbazole compounds in Clausena excavata by RP-HPLCKongkathip B., Sutthiprabha S., Yoosook C., Mongkolsook Y., Kongkathip N.2010Journal of Chromatographic Science
    48(6),pp. 445-449
    7
    26Synthesis and anticancer evaluation of naphthoquinone esters with 2′-cyclopentyl and 2′-cyclohexyl substituentsKongkathip N., Pradidphol N., Hasitapan K., Kongkathip B.2010Bioscience, Biotechnology and Biochemistry
    74(6),pp. 1205-1214
    7
    27Total synthesis of (+)-epiquinamide and (−)-epiepiquinamide from D-mannoseSangsuwan W., Kongkathip B., Chuawong P., Kongkathip N.2017Tetrahedron
    73(52),pp. 7274-7281
    7
    28Biophysical and molecular docking studies of naphthoquinone derivatives on the ATPase domain of human Topoisomerase IIBoonyalai N., Sittikul P., Pradidphol N., Kongkathip N.2013Biomedicine and Pharmacotherapy
    67(2),pp. 122-128
    7
    29Biosynthetic origins of menisporopsin AWattana-Amorn P., Juthaphan P., Sirikamonsil M., Sriboonlert A., Simpson T., Kongkathip N.2013Journal of Natural Products
    76(7),pp. 1235-1237
    6
    30Identification of Saccharomyces cerevisiae Tub1 α-tubulin as a potential target for NKH-7, a cytotoxic 1-naphthol derivative compoundChanklan R., Chanklan R., Mizunuma M., Kongkathip N., Hasitapan K., Kongkathip B., Miyakawa T.2008Bioscience, Biotechnology and Biochemistry
    72(4),pp. 1023-1031
    5
    31New strategy for synthesis of the disaccharide moiety of the highly potent anticancer natural product OSW-1Kongkathip B., Kongkathip N., Rujirawanich J.2014Synthetic Communications
    44(15),pp. 2248-2255
    4
    32Synthesis of novel 2-(2′-cyclopentyl)- and 2-(2′-cyclohexyl) substituted 1-naphthol derivatives with anticyclooxygenase activityKongkathip N., Hasitapan K., Pradidphol N., Kirtikara K., Jongkon N., Kongkathip B.2006Current Medicinal Chemistry
    13(30),pp. 3663-3674
    4
    33Syntheses of both diastereoisomers of 2,8-dioxabicyclo[3.2.1]octane derivatives: Degradation products of Daphniphyllum alkaloidsKongkathip B., Sookkho R., Kongkathip N., Taylor W.C.1999Chemistry Letters
    (10),pp. 1095-1096
    4
    34Simple and convenient method for the synthesis of Δ9(11)-3-hydroxy, Δ1,4- and Δ1,4,9(11)-3-ketosteroids by selective dehydrogenation of 3-hydroxy-12-ketosteroidsKongkathip B., Kongkathip N., Khunnavutimanotum P., Sakee U.1998Chemistry Letters
    (12),pp. 1207-1208
    3
    35In vitro and in silico studies of naphthoquinones and peptidomimetics toward Plasmodium falciparum plasmepsin VSittikul P., Sittikul P., Songtawee N., Kongkathip N., Boonyalai N., Boonyalai N.2018Biochimie
    152,pp. 159-173
    3
    36A new approach to asymmetric synthesis of (−)-epiquinamide from D-glucoseLumyong K., Kongkathip B., Chuanopparat N., Kongkathip N.2019Tetrahedron
    75(4),pp. 533-537
    3
    37Synthesis of N-formylnornuciferine with cardiotonic activityImphanban K., Kongkathip N., Dhumma-upakorn P., Mesripong R., Kongkathip B.2009Kasetsart Journal - Natural Science
    43(4),pp. 738-744
    2
    38An efficient synthesis and regioselective hydrogenolysis of dioxolane-type of carbohydratesKongkathip B., Chuanopparat N., Kongkathip N.2016Tetrahedron
    72(23),pp. 3296-3304
    1
    39Erratum: Palladium catalysed reactions of allene with active methylene pronucleophiles. C-1,3-Dienylmethyl derivatives and their Diels-Alder reactions (Tetrahedron (2001) 57 (9187-9197) PII: S0040402001009243)Grigg R., Kongkathip N., Kongkathip B., Luangkamin S., Dondas H.A.2002Tetrahedron
    58(2),pp. 377
    1
    40Efficient synthesis of 16α-methyl cyproterone acetateSakee U., Kongkathip B., Kongkathip N.2003Journal of Chemical Research - Part S
    (1),pp. 12-13
    1
    41The first syntheses of 16β-chloro- and 16β-bromo-cyproterone acetateSakee U., Kongkathip N., Kongkathip B.2003Synthetic Communications
    33(10),pp. 1695-1706
    1
    42Synthesis and cytotoxicity studies of polyhydroxysterols and their sulfate analogsBunyathaworn P., Kongkathip B., Kongkathip N.2011Kasetsart Journal - Natural Science
    45(4),pp. 700-716
    0
    43Synthesis and biological evaluation of 3,16,20-polyoxygenated steroids of marine origin and their analogsBoonananwong S., Kongkathip B., Kongkathip N.2008Kasetsart Journal - Natural Science
    42(3),pp. 531-542
    0
    44A quick and convenient 1H quantitative NMR method for determination of bioactive pyranocoumarins from Clausena excavataSakarat N., Prapapongpan P., Prapapongpan P., Sae-Lim S., Saleepochn T., Kongkathip B., Kongkathip N., Yakhampom S., Wongprom J., Chuawong P.2021Phytochemistry Letters
    45,pp. 126-131
    0
    45Potent antitumor activity of synthetic 1,2-naphthoquinones and 1,4-naphthoquinonesKongkathip N., Kongkathip B., Siripong P., Sangma C., Luangkamin S., Niyomdecha M., Pattanapa S., Piyaviriyagul S., Kongsaeree P.2003Bioorganic and Medicinal Chemistry
    11(14),pp. 3179-3191
    194
    46Coumarins and carbazoles from Clausena excavata exhibited antimycobacterial and antifungal activitiesSunthitikawinsakul A., Kongkathip N., Kongkathip B., Phonnakhu S., Daly J., Spande T., Nimit Y., Rochanaruangrai S.2003Planta Medica
    69(2),pp. 155-157
    124
    47Anti-HIV-1 constituents from Clausena excavata: Part II. Carbazoles and a pyranocoumarinKongkathip B., Kongkathip N., Sunthitikawinsakul A., Napaswat C., Yoosook C.2005Phytotherapy Research
    19(8),pp. 728-731
    86
    48Stereoselective palladium-catalyzed four-component cascade synthesis of pyrrolidinyl-, pyrazolidinyl-, and isoxazolidinyl isoquinolinesDondas H., Dondas H., Fishwick C., Gai X., Grigg R., Kilner C., Dumrongchai N., Kongkathip B., Kongkathip N., Polysuk C., Sridharan V.2005Angewandte Chemie - International Edition
    44(46),pp. 7570-7574
    63
    49Synthesis of novel rhinacanthins and related anticancer naphthoquinone estersKongkathip N., Luangkamin S., Kongkathip B., Sangma C., Grigg R., Kongsaeree P., Prabpai S., Pradidphol N., Piyaviriyagul S., Siripong P.2004Journal of Medicinal Chemistry
    47(18),pp. 4427-4438
    59
    50Biologically active substances from amphibians: Preliminary studies on anurans from twenty-one genera of ThailandDaly J.W., Noimai N., Kongkathip B., Kongkathip N., Wilham J.M., Garraffo H.M., Kaneko T., Spande T.F., Nimit Y., Nabhitabhata J., Chan-Ard T.2004Toxicon
    44(8),pp. 805-815
    57
    51Antimicrobial activity of curcuminoids from Curcuma Longa L. on pathogenic bacteria of shrimp and chickenLawhavinit O., Kongkathip N., Kongkathip B.2010Kasetsart Journal - Natural Science
    44(3),pp. 364-371
    39
    52Study on cardiac contractility of cycloeucalenol and cycloeucalenone isolated from Tinospora crispaKongkathip N., Dhumma-upakorn P., Kongkathip B., Chawananoraset K., Sangchomkaeo P., Hatthakitpanichakul S.2002Journal of Ethnopharmacology
    83(1-2),pp. 95-99
    38
    53Anti-HIV-1 Limonoid: First Isolation from Clausena excavataSunthitikawinsakul A., Kongkathip N., Kongkathip B., Phonnakhu S., Daly J., Spande T., Nimit Y., Napaswat C., Kasisit J., Yoosook C.2003Phytotherapy Research
    17(9),pp. 1101-1103
    37
    54First synthesis and anticancer activity of novel naphthoquinone amidesPradidphol N., Kongkathip N., Sittikul P., Boonyalai N., Kongkathip B.2012European Journal of Medicinal Chemistry
    49,pp. 253-270
    34
    55Induction of apoptosis by rhinacanthone isolated from Rhinacanthus nasutus roots in human cervical carcinoma cellsSiripong P., Hahnvajanawong C., Yahuafai J., Piyaviriyakul S., Piyaviriyakul S., Kanokmedhakul K., Kongkathip N., Ruchirawat S., Oku N.2009Biological and Pharmaceutical Bulletin
    32(7),pp. 1251-1260
    33
    56An efficient synthesis of oseltamivir phosphate (Tamiflu) via a metal-mediated domino reaction and ring-closing metathesisWichienukul P., Akkarasamiyo S., Kongkathip N., Kongkathip B.2010Tetrahedron Letters
    51(24),pp. 3208-3210
    32
    57Constituents and bioactivities of Clausena excavataKongkathip N., Kongkathip B.2009Heterocycles
    79(C),pp. 121-144
    31